|
Bromodomains
AMSBIO supplies a unique range of products for bromodomain research. Bromodomains are protein domains that recognise acetylated lysine. They are implicated in cancer, obesity, inflammation and diabetes. They play an important role in epigenetics.
AMSBIO provides an ever-growing portfolio of BRDs and kits suitable for bromodomain profiling, inhibitor screening assays, and drug discovery.
Inhibitor screening assays
The Inhibitor Screening Assay Kits are designed to measure the inhibition of bromodomain protein binding to its substrate. The key to the Assay Kits is the highly specific binding of the bromodomains to the acetylated histone substrate.
Homogenous assays
The TR-FRET Assay Kits are designed to measure the inhibition of protein binding to its substrate in a homogeneous 384 reaction format. This FRET-based assay requires no time-consuming washing steps, making it especially suitable for high throughput screening applications. The assay procedure is straightforward and simple.
BRD Proteins
Product list:
31025
|
BRD2 (BD1+BD2), His-tag
|
100 ug
|
|
31045
|
BRD4 (BD1+BD2), His-tag
|
100 ug
|
|
31119
|
CREBBP (KAT3A), His-tag
|
100 ug
|
|
31118
|
P300 (1046-1163), His-tag
|
100 ug
|
|
31060
|
BRDT (BD2), GST-tag
|
100 ug
|
|
31061
|
BRDT (BD1+BD2), GST-tag
|
100 ug
|
|
31123
|
TAF1 (BD1), His-tag
|
100 ug
|
|
31034
|
BRD3 (BD1+BD2), His-tag
|
100 ug
|
|
31035
|
BRD3 (BD1+BD2), GST-tag
|
100 ug
|
|
31124
|
TAF1 (BD1+BD2), GST-tag
|
100 ug
|
|
31126
|
TAF1 (BD2), GST-tag
|
100 ug
|
|
31031
|
BRD3 (BD2), His-tag
|
100 ug
|
|
31033
|
BRD3 (BD2), GST-tag
|
100 ug
|
|
31030
|
BRD3 (BD1), His-tag
|
100 ug
|
|
31032
|
BRD3 (BD1), GST-tag
|
100 ug
|
|
31020
|
BRD2 (BD2), His-tag
|
100 ug
|
|
31022
|
BRD2 (BD1), His-tag
|
100 ug
|
|
31021
|
BRD2 (BD1), GST-tag
|
100 ug
|
|
31023
|
BRD2 (BD2), GST-tag
|
100 ug
|
|
31010
|
BRD1, His-tag
|
100 ug
|
|
31040
|
BRD4 (BD1), GST-tag
|
100 ug
|
|
31041
|
BRD4 (BD2), GST-tag
|
100 ug
|
|
31102
|
SMARCA4 (BRG1), His-tag
|
100 ug
|
|
31043
|
BRD4 (BD2), His-tag
|
100 ug
|
|
31104
|
TAF1L (BD2), His-tag
|
100 ug
|
|
31101
|
BRDT (BD1), His-tag
|
100 ug
|
|
31042
|
BRD4 (BD1), His-tag
|
100 ug
|
|
31103
|
TAF1L (BD1), His-tag
|
100 ug
|
|
31100
|
BRDT (BD2), His-tag
|
100 ug
|
|
31090
|
BRD9, His-tag
|
100 ug
|
|
31105
|
TAF1L (BD1), GST-tag
|
100 ug
|
|
31106
|
TAF1L (BD2), GST-tag
|
100 ug
|
|
31107
|
TAF1L (BD1+BD2), GST-tag
|
100 ug
|
|
31024
|
BRD2 (BD1+BD2), GST-tag
|
100 ug
|
|
31011
|
BRD1, GST-tag
|
100 ug
|
|
31108
|
BRDT (BD1), GST-tag
|
100 ug
|
|
31109
|
ATAD2A, His-tag
|
100 ug
|
|
31110
|
TAF1 (BD2), His-tag
|
100 ug
|
|
31111
|
SMARCA2, His-tag
|
100 ug
|
|
31113
|
BAZ2B, His-tag
|
100 ug
|
|
31112
|
BRPF1, His-tag
|
100 ug
|
|
31114
|
GCN5 (727-837), His-tag
|
100 ug
|
|
31115
|
WDR9/BRWD1 (BD2), His-tag
|
100 ug
|
|
31116
|
TRIM24 (TIF1), His-tag
|
100 ug
|
|
31125
|
ATAD2B (KIAA1240), GST-tag
|
100 ug
|
|
31117
|
ATAD2B (KIAA1240), His-tag
|
100 ug
|
|
31044
|
BRD4 (BD1+BD2), GST-tag
|
100 ug
|
|
31122
|
PB1 (BD4), His-tag
|
100 ug
|
|
31120
|
PCAF (KAT2B), His-tag
|
100 ug
|
|
31121
|
ATAD2A, GST-tag
|
100 ug
|
|
31141
|
SMARCA2, GST-tag
|
100 ug
|
|
31133
|
PB1 (BD6), His-tag
|
100 ug
|
|
31131
|
FALZ (BPTF), His-tag
|
100 ug
|
|
31046
|
CECR2, His-tag
|
100 ug
|
|
31130
|
BRPF3, GST-tag
|
100 ug
|
|
31047
|
BRD4 (BD1+BD2)
|
100 ug
|
|
31132
|
SMARCA4 (BRG1), GST-tag
|
100 ug
|
|
31137
|
BAZ1B, GST-tag
|
100 ug
|
|
31145
|
BAZ1B, His-tag
|
100 ug
|
|
31144
|
ZMYND11, GST-tag
|
100 ug
|
|
31147
|
ASH1L, His-tag
|
100 ug
|
|
31146
|
TRIM28, His-tag
|
100 ug
|
|
31143
|
ZMYND8, GST-tag
|
100 ug
|
|
31142
|
PHIP (BD1), GST-tag
|
100 ug
|
|
31140
|
PHIP (BD1), His-tag
|
100 ug
|
|
31139
|
TRIM28, GST-tag
|
100 ug
|
|
31138
|
CECR2, GST-tag
|
100 ug
|
|
31136
|
BAZ1A, GST-tag
|
100 ug
|
|
31135
|
WDR9/BRWD1 (BD2), GST-tag
|
100 ug
|
|
31134
|
FALZ (BPTF), GST-tag
|
100 ug
|
|
31128
|
CREBBP (KAT3A), GST-tag
|
100 ug
|
|
31127
|
TRIM24 (TIF1), GST-tag
|
100 ug
|
|
31091
|
BRD9, GST-tag
|
100 ug
|
|
| | | |
|